Zacopride hydrochloride
CAS No. 101303-98-4
Zacopride hydrochloride ( —— )
产品货号. M20083 CAS No. 101303-98-4
Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥721 | 有现货 |
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10MG | ¥1191 | 有现货 |
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25MG | ¥2406 | 有现货 |
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50MG | ¥3872 | 有现货 |
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100MG | ¥5581 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Zacopride hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
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产品描述Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT3 antagonist; 5-HT4 agonist; IK1/Kir2.1 agonist
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研究领域——
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适应症——
化学信息
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CAS Number101303-98-4
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分子量346.26
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分子式C15H20ClN3O2.HCl
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纯度>98% (HPLC)
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溶解度DMSO:10 mM
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SMILESCl.COc1cc(N)c(Cl)cc1C(=O)NC1CN2CCC1CC2
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Nagakura Y et al. Pharmacological properties of a novel gastrointestinal prokinetic benzamide selective for human 5-HT4 receptor versus human 5-HT3 receptor. Pharmacol Res. 1999 May;39(5):375-82.
产品手册
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